Heitmann T, Liao G, Ernst G, Poslusney M, van Kralingen T, Li Y, Masi M, DePasquale M, Buchler I, Wei H, Carr GV, Shlevkov E, Lu M, Jessen H, Barrow JC., 2024, Identification and Characterization of a Blood-Brain Barrier Penetrant Inositol Hexakisphosphate Kinase (IP6K) Inhibitor, J Med Chem., 67(16):13639-13665. doi: 10.1021/acs.jmedchem.4c00190. PMID: 39096294 PubMed
Heitmann T, Liao G, de León P, Ernst G, Buchler I, Wei H, Shlevkov E, Brown D, Fitzek M, Collier M, Smith DM, Barrow JC., 2023, Fragment-Based Screening Identifies New Quinazolinone-Based Inositol Hexakisphosphate Kinase (IP6K) Inhibitors, ACS Med Chem Lett., 14(12):1760-1766. doi: 10.1021/acsmedchemlett.3c00409. PMCID: PMC10726443 PubMed
Heitmann T, Barrow JC., 2023, The Role of Inositol Hexakisphosphate Kinase in the Central Nervous System, Biomolecules, 13(9):1317. doi: 10.3390/biom13091317. PMCID: PMC10526494 PubMed